标题
Late-stage [18F]fluorination: new solutions to old problems
作者
关键词
-
出版物
Chemical Science
Volume 5, Issue 12, Pages 4545-4553
出版商
Royal Society of Chemistry (RSC)
发表日期
2014-08-25
DOI
10.1039/c4sc02099e
参考文献
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注意:仅列出部分参考文献,下载原文获取全部文献信息。- PET Project
- (2015) CHEMICAL & ENGINEERING NEWS
- High Affinity Radiopharmaceuticals Based Upon Lansoprazole for PET Imaging of Aggregated Tau in Alzheimer’s Disease and Progressive Supranuclear Palsy: Synthesis, Preclinical Evaluation, and Lead Selection
- (2014) Maria V. Fawaz et al. ACS Chemical Neuroscience
- Synthesis and Imaging Validation of [18F]MDL100907 Enabled by Ni-Mediated Fluorination
- (2014) Hong Ren et al. ACS Chemical Neuroscience
- A General Copper-Mediated Nucleophilic18F Fluorination of Arenes
- (2014) Matthew Tredwell et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- A Universal Procedure for the [18F]Trifluoromethylation of Aryl Iodides and Aryl Boronic Acids with Highly Improved Specific Activity
- (2014) Dion van der Born et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Cu(i)-mediated 18F-trifluoromethylation of arenes: Rapid synthesis of 18F-labeled trifluoromethyl arenes
- (2014) T. Rühl et al. CHEMICAL COMMUNICATIONS
- [18F]CuCF3: A [18F]Trifluoromethylating Agent for Arylboronic Acids and Aryl Iodides
- (2014) Pavel Ivashkin et al. CHEMISTRY-A EUROPEAN JOURNAL
- Radiosyntheses using Fluorine-18: The Art and Science of Late Stage Fluorination
- (2014) Erin Cole et al. CURRENT TOPICS IN MEDICINAL CHEMISTRY
- Regulatory Requirements for PET Drug Production
- (2014) S. W. Schwarz et al. JOURNAL OF NUCLEAR MEDICINE
- Enantioselective Radiosynthesis of Positron Emission Tomography (PET) Tracers Containing [18F]Fluorohydrins
- (2014) Thomas J. A. Graham et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Late Stage Benzylic C–H Fluorination with [18F]Fluoride for PET Imaging
- (2014) Xiongyi Huang et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Copper-Catalyzed [18F]Fluorination of (Mesityl)(aryl)iodonium Salts
- (2014) Naoko Ichiishi et al. ORGANIC LETTERS
- Spirocyclic hypervalent iodine(III)-mediated radiofluorination of non-activated and hindered aromatics
- (2014) Benjamin H. Rotstein et al. Nature Communications
- Iodonium ylides for one-step, no-carrier-added radiofluorination of electron rich arenes, exemplified with 4-(([18F]fluorophenoxy)-phenylmethyl)piperidine NET and SERT ligands
- (2014) Jens Cardinale et al. RSC Advances
- Synthesis, 18F-Radiolabeling, and in Vivo Biodistribution Studies of N-Fluorohydroxybutyl Isatin Sulfonamides using Positron Emission Tomography
- (2013) Panupun Limpachayaporn et al. JOURNAL OF MEDICINAL CHEMISTRY
- Novel 18F-Labeled Arylquinoline Derivatives for Noninvasive Imaging of Tau Pathology in Alzheimer Disease
- (2013) N. Okamura et al. JOURNAL OF NUCLEAR MEDICINE
- Cu(OTf)2-Mediated Fluorination of Aryltrifluoroborates with Potassium Fluoride
- (2013) Yingda Ye et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- A broadly applicable [18F]trifluoromethylation of aryl and heteroaryl iodides for PET imaging
- (2013) Mickael Huiban et al. Nature Chemistry
- Cu-Catalyzed Fluorination of Diaryliodonium Salts with KF
- (2013) Naoko Ichiishi et al. ORGANIC LETTERS
- Application of Palladium-Mediated 18F-Fluorination to PET Radiotracer Development: Overcoming Hurdles to Translation
- (2013) Adam S. Kamlet et al. PLoS One
- Mechanism of electrophilic fluorination with Pd(iv): fluoride capture and subsequent oxidative fluoride transfer
- (2013) Jochen R. Brandt et al. Chemical Science
- 18F Labeling of Arenes
- (2012) Matthew Tredwell et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Metal-Free Oxidative Fluorination of Phenols with [18F]Fluoride
- (2012) Zhanghua Gao et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Nickel-Mediated Oxidative Fluorination for PET with Aqueous [18F] Fluoride
- (2012) Eunsung Lee et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Direct, nucleophilic radiosynthesis of [18F]trifluoroalkyl tosylates: improved labelling procedures
- (2012) Patrick J. Riss et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Regio- and stereoretentive synthesis of branched, linear (E)- and (Z)-allyl fluorides from allyl carbonates under Ir-catalysis
- (2012) Elena Benedetto et al. Chemical Science
- Positron emission tomography molecular imaging for drug development
- (2011) Paul M. Matthews et al. BRITISH JOURNAL OF CLINICAL PHARMACOLOGY
- A simple, rapid procedure for nucleophilic radiosynthesis of aliphatic [18F]trifluoromethyl groups
- (2011) Patrick J. Riss et al. CHEMICAL COMMUNICATIONS
- Rapid and Efficient Radiosyntheses of meta-Substituted [18F]Fluoroarenes from [18F]Fluoride Ion and Diaryliodonium Tosylates within a Microreactor
- (2011) Joong-Hyun Chun et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- Iridium-Catalyzed Allylic Fluorination of Trichloroacetimidates
- (2011) Joseph J. Topczewski et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- A Fluoride-Derived Electrophilic Late-Stage Fluorination Reagent for PET Imaging
- (2011) E. Lee et al. SCIENCE
- PET radiotracers: crossing the blood–brain barrier and surviving metabolism
- (2009) Victor W. Pike TRENDS IN PHARMACOLOGICAL SCIENCES
- Molecular Imaging with PET
- (2008) Simon M. Ametamey et al. CHEMICAL REVIEWS
- Chemistry with [18F]Fluoride Ion
- (2008) Lisheng Cai et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- Synthesis, radiofluorination and first evaluation of (±)-[18F]MDL 100907 as serotonin 5-HT2Areceptor antagonist for PET
- (2008) Ute Mühlhausen et al. JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS
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