期刊
SYNLETT
卷 -, 期 17, 页码 2511-2515出版社
GEORG THIEME VERLAG KG
DOI: 10.1055/s-0032-1317320
关键词
cascade synthesis; 2-substituted indoles; palladium-catalyzed; cross-coupling reaction
An efficient cascade methodology toward the synthesis of 2-substituted indoles has been developed. The transformation proceeds via a palladium-catalyzed cross-coupling reaction of o-nitrobenzyl cyanides with boronic acids. The use of Fe as co-catalyst during the course of reaction employs significant enhancement in reaction rates. The developed protocol allows for the unprecedented use of arylboronic acids as coupling partners for constructing 2-substituted indoles.
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