The synthesis and preclinical evaluation in rhesus monkey of [18F]MK-6577 and [11C]CMPyPB glycine transporter 1 positron emission tomography radiotracers

Identification and evaluation of [11C]GSK931145 as a novel ligand for imaging the type 1 glycine transporter with positron emission tomography

(2010) J. Passchier et al.   SYNAPSE

Discovery of N-{[1-(propylsulfonyl)-4-pyridin-2-ylpiperidin-4-yl]methyl}benzamides as novel, selective and potent GlyT1 inhibitors

(2009) Zhijian Zhao et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Discovery of GlyT1 inhibitors with improved pharmacokinetic properties

(2009) Scott E. Wolkenberg et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Optimisation of a series of potent, selective and orally bioavailable GlyT1 inhibitors

(2009) Joanne L. Thomson et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Inverse agonist histamine H3 receptor PET tracers labelled with carbon-11 or fluorine-18

(2009) Terence G. Hamill et al.   SYNAPSE

[11C]GSK931145: A new pet ligand for glycine transporter 1

(2008) N. Venkatesha Murthy et al.   NEUROIMAGE

A novel radioligand for glycine transporter 1: characterization and use in autoradiographic and in vivo brain occupancy studies

(2008) Zhizhen Zeng et al.   NUCLEAR MEDICINE AND BIOLOGY