Blockade of the brain histamine H3 receptor by JNJ-39220675: preclinical PET studies with [11C]GSK189254 in anesthetized baboon

Pre-clinical characterization of aryloxypyridine amides as histamine H3 receptor antagonists: Identification of candidates for clinical development

(2010) Michael A. Letavic et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Evaluation of 11C-GSK189254 as a Novel Radioligand for the H3 Receptor in Humans Using PET

(2010) S. Ashworth et al.   JOURNAL OF NUCLEAR MEDICINE

Histamine and H3 Receptor in Alcohol-Related Behaviors

(2010) P. Panula et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

The Histamine H3 Receptor and Eating Behavior

(2010) M. B. Passani et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

JNJ-39220675, a novel selective histamine H3 receptor antagonist, reduces the abuse-related effects of alcohol in rats

(2010) Ruggero Galici et al.   PSYCHOPHARMACOLOGY

Effects of Modafinil on Dopamine and Dopamine Transporters in the Male Human Brain

(2009) Nora D. Volkow et al.   JAMA-JOURNAL OF THE AMERICAN MEDICAL ASSOCIATION

Measuring Drug Occupancy in the Absence of a Reference Region: The Lassen Plot Re-Visited

(2009) Vincent J Cunningham et al.   JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM

11C-GSK189254: A Selective Radioligand for In Vivo Central Nervous System Imaging of Histamine H3 Receptors by PET

(2009) C. Plisson et al.   JOURNAL OF NUCLEAR MEDICINE

Reversible Inhibitors of Monoamine Oxidase-A (RIMAs): Robust, Reversible Inhibition of Human Brain MAO-A by CX157

(2009) Joanna S Fowler et al.   NEUROPSYCHOPHARMACOLOGY

2-Aryloxymethylmorpholine histamine H3 antagonists

(2008) Michael A. Letavic et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

The histamine H3receptor: an attractive target for the treatment of cognitive disorders

(2008) T A Esbenshade et al.   BRITISH JOURNAL OF PHARMACOLOGY