FRET-Based Detection of M1 Muscarinic Acetylcholine Receptor Activation by Orthosteric and Allosteric Agonists

Helix 8 of the M1 Muscarinic Acetylcholine Receptor: Scanning Mutagenesis Delineates a G Protein Recognition Site

(2011) R. G. Kaye et al.   MOLECULAR PHARMACOLOGY

FRET-based sensors for the human M1-, M3-, and M5-acetylcholine receptors

(2010) Nicole Ziegler et al.   BIOORGANIC & MEDICINAL CHEMISTRY

A Fluorescence Resonance Energy Transfer-based M2Muscarinic Receptor Sensor Reveals Rapid Kinetics of Allosteric Modulation

(2010) Monika Maier-Peuschel et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Kinetics of M1muscarinic receptor and G protein signaling to phospholipase C in living cells

(2010) Björn H. Falkenburger et al.   JOURNAL OF GENERAL PHYSIOLOGY

Mechanical stimulus alters conformation of type 1 parathyroid hormone receptor in bone cells

(2009) Yan-Liang Zhang et al.   AMERICAN JOURNAL OF PHYSIOLOGY-CELL PHYSIOLOGY

Fluorescence changes reveal kinetic steps of muscarinic receptor–mediated modulation of phosphoinositides and Kv7.2/7.3 K+channels

(2009) Jill B. Jensen et al.   JOURNAL OF GENERAL PHYSIOLOGY

Subtype-selective allosteric modulators of muscarinic receptors for the treatment of CNS disorders

(2009) P. Jeffrey Conn et al.   TRENDS IN PHARMACOLOGICAL SCIENCES

Characterization of a CNS penetrant, selective M1muscarinic receptor agonist, 77-LH-28-1

(2008) C J Langmead et al.   BRITISH JOURNAL OF PHARMACOLOGY

Dual Role of the β2-Adrenergic Receptor C Terminus for the Binding of β-Arrestin and Receptor Internalization

(2008) Cornelius Krasel et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

G Protein Coupling and Signaling Pathway Activation by M1 Muscarinic Acetylcholine Receptor Orthosteric and Allosteric Agonists

(2008) R. L. Thomas et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

Mutagenic Mapping Suggests a Novel Binding Mode for Selective Agonists of M1 Muscarinic Acetylcholine Receptors

(2008) G. Lebon et al.   MOLECULAR PHARMACOLOGY

Fluorescence Resonance Energy Transfer Analysis of  2a-Adrenergic Receptor Activation Reveals Distinct Agonist-Specific Conformational Changes

(2008) A. Zurn et al.   MOLECULAR PHARMACOLOGY

Discovery and Characterization of Novel Allosteric Potentiators of M1 Muscarinic Receptors Reveals Multiple Modes of Activity

(2008) J. E. Marlo et al.   MOLECULAR PHARMACOLOGY

Optical techniques to analyze real-time activation and signaling of G-protein-coupled receptors

(2008) Martin J. Lohse et al.   TRENDS IN PHARMACOLOGICAL SCIENCES

Intracellular Mechanisms Regulating Corticotropin-Releasing Hormone Receptor-2β Endocytosis and Interaction with Extracellularly Regulated Kinase 1/2 and p38 Mitogen-Activated Protein Kinase Signaling Cascades

(2007) Danijela Markovic et al.   MOLECULAR ENDOCRINOLOGY

Muscarinic acetylcholine receptors as CNS drug targets

(2007) Christopher J. Langmead et al.   PHARMACOLOGY & THERAPEUTICS