期刊
ORGANIC LETTERS
卷 14, 期 14, 页码 3800-3803出版社
AMER CHEMICAL SOC
DOI: 10.1021/ol301700y
关键词
-
资金
- National Institutes of Health [GM58160, F32GM097771]
- Amgen
- National Science Foundation [CHE-9808061]
A method for the Pd-catalyzed N-arylation of both aryl and alkyl amidines with a wide range of aryl bromides, chlorides, and triflates is described. The reactions proceed in short reaction times and with excellent selectivity for monoarylation. A one-pot synthesis of quinazoline derivatives, via addition of an aldehyde to the crude reaction mixture following Pd-catalyzed N-arylation, is also demonstrated.
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