Design, physico-chemical and pre-clinical evaluation of a homo-bivalent 99mTc-(BTZ)2DTPA radioligand for targeting dimeric 5-HT1A/5-HT7 receptors

Mapping neuroreceptors with metal-labeled radiopharmaceuticals

(2017) S. Chaturvedi et al.   MedChemComm

Structural basis to characterise transactivation domain of BRCA1

(2016) Lumbini R. Yadav et al.   JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS

Folate-conjugated polyspermine for lung cancer–targeted gene therapy

(2016) Mei Zhang et al.   Acta Pharmaceutica Sinica B

The 5-HT7 receptor as a potential target for treating drug and alcohol abuse

(2015) Sheketha R. Hauser et al.   Frontiers in Neuroscience

Interplay between Serotonin 5-HT1Aand 5-HT7Receptors in Depressive Disorders

(2014) Vladimir S. Naumenko et al.   CNS Neuroscience & Therapeutics

Structure–activity relationships and molecular modeling studies of novel arylpiperazinylalkyl 2-benzoxazolones and 2-benzothiazolones as 5-HT7 and 5-HT1A receptor ligands

(2014) Loredana Salerno et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Fluoridonitrosyl Complexes of Technetium(I) and Technetium(II). Synthesis, Characterization, Reactions, and DFT Calculations

(2014) Samundeeswari Mariappan Balasekaran et al.   INORGANIC CHEMISTRY

Design, synthesis and preliminary evaluation of a novel SPECT DTPA-bis-triazaspirodecanone conjugate for D2receptor imaging

(2014) Swarndeep K. Sethi et al.   RSC Advances

Smart polymers for the controlled delivery of drugs – a concise overview

(2014) Honey Priya James et al.   Acta Pharmaceutica Sinica B

Bivalent Ligands That Target μ Opioid (MOP) and Cannabinoid1 (CB1) Receptors Are Potent Analgesics Devoid of Tolerance

(2013) Morgan Le Naour et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis, docking and preliminary in vivo evaluation of serotonin dithiocarbamate as novel SPECT neuroimaging agent

(2013) Shubhra Chaturvedi et al.   MedChemComm

Major channels involved in neuropsychiatric disorders and therapeutic perspectives

(2013) Paola Imbrici et al.   Frontiers in Genetics

Influence of Spacer–Receptor Interactions on the Stability of Bivalent Ligand–Receptor Complexes

(2012) Jorge Numata et al.   JOURNAL OF PHYSICAL CHEMISTRY B

Neurotransmitter receptors and cognitive dysfunction in Alzheimer's disease and Parkinson's disease

(2012) Yunqi Xu et al.   PROGRESS IN NEUROBIOLOGY

Bridging the gap: bitopic ligands of G-protein-coupled receptors

(2012) J. Robert Lane et al.   TRENDS IN PHARMACOLOGICAL SCIENCES

A homodimeric bivalent radioligand derived from 1-(2-methoxyphenyl)piperazine with high affinity for in vivo 5-HT1A receptor imaging

(2012) Niraj Singh et al.   MedChemComm

Bivalent Dopamine D2Receptor Ligands: Synthesis and Binding Properties

(2011) Julia Kühhorn et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of Specific SPECT-Radiopharmaceutical for Tumor Imaging Based on Methionine:99mTc-DTPA-bis(methionine)

(2010) Puja Panwar Hazari et al.   BIOCONJUGATE CHEMISTRY

Discovery of Bishomo(hetero)arylpiperazines as Novel Multifunctional Ligands Targeting Dopamine D3and Serotonin 5-HT1Aand 5-HT2AReceptors

(2010) Stefania Butini et al.   JOURNAL OF MEDICINAL CHEMISTRY

Bivalent Ligands of CXCR4 with Rigid Linkers for Elucidation of the Dimerization State in Cells

(2010) Tomohiro Tanaka et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Thermodynamics of Multivalent Interactions: Influence of the Linker

(2010) Ravi S. Kane   LANGMUIR

Molecular modeling of the human serotonin1Areceptor: role of membrane cholesterol in ligand binding of the receptor

(2010) Yamuna Devi Paila et al.   Molecular BioSystems

Serotonin 5-HT7 receptor agents: Structure-activity relationships and potential therapeutic applications in central nervous system disorders

(2010) Marcello Leopoldo et al.   PHARMACOLOGY & THERAPEUTICS

Nanoparticle interaction with plasma proteins as it relates to particle biodistribution, biocompatibility and therapeutic efficacy

(2009) Parag Aggarwal et al.   ADVANCED DRUG DELIVERY REVIEWS

Rational Design of Amyloid Binding Agents Based on the Molecular Rotor Motif

(2009) Jeyanthy Sutharsan et al.   ChemMedChem

1,1′-Disubstituted Ferrocenes as Molecular Hinges in Mono- and Bivalent Dopamine Receptor Ligands

(2009) Daniela Huber et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of New Serotonin 5-HT7Receptor Ligands. Determinants of 5-HT7/5-HT1AReceptor Selectivity

(2009) Rocío A. Medina et al.   JOURNAL OF MEDICINAL CHEMISTRY

Adenosine A2AReceptor-Antagonist/Dopamine D2Receptor-Agonist Bivalent Ligands as Pharmacological Tools to Detect A2A-D2Receptor Heteromers

(2009) Aroa Soriano et al.   JOURNAL OF MEDICINAL CHEMISTRY

Serotonin Receptors

(2008) David E. Nichols et al.   CHEMICAL REVIEWS

Synthesis of New Arylpiperazinylalkylthiobenzimidazole, Benzothiazole, or Benzoxazole Derivatives as Potent and Selective 5-HT1ASerotonin Receptor Ligands†

(2008) Maria A. Siracusa et al.   JOURNAL OF MEDICINAL CHEMISTRY