Catalyst-free synthesis of quinazolin-4-ones from (hetero)aryl-guanidines: application to the synthesis of pyrazolo[4,3-f]quinazolin-9-ones, a new family of DYRK1A inhibitors

Synthesis and SAR of new pyrazolo[4,3-h]quinazoline-3-carboxamide derivatives as potent and selective MPS1 kinase inhibitors

(2011) Marina Caldarelli et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and biological evaluation of new 3-(6-hydroxyindol-2-yl)-5-(Phenyl) pyridine or pyrazine V-Shaped molecules as kinase inhibitors and cytotoxic agents

(2011) Pamela Kassis et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Leucettines, a Class of Potent Inhibitors of cdc2-Like Kinases and Dual Specificity, Tyrosine Phosphorylation Regulated Kinases Derived from the Marine Sponge Leucettamine B: Modulation of Alternative Pre-RNA Splicing

(2011) Mansour Debdab et al.   JOURNAL OF MEDICINAL CHEMISTRY

β-Carboline Compounds, Including Harmine, Inhibit DYRK1A and Tau Phosphorylation at Multiple Alzheimer's Disease-Related Sites

(2011) Danielle Frost et al.   PLoS One

Montmorillonite K-10 catalyzed cyclization of N-ethoxycarbonyl-N′-arylguanidines: Access to pyrimido[4,5-c]carbazole and pyrimido[5,4-b]indole derivatives

(2010) Julien Debray et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Swift and Efficient Synthesis of 4-Phenylquinazolines: Involvement ofN-Heterocyclic Carbene in the Key Cyclization Step

(2010) Julien Debray et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and biological evaluation of 3,6-diamino-1H-pyrazolo[3,4-b]pyridine derivatives as protein kinase inhibitors

(2009) Mourad Chioua et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Evaluation of substituted 6-arylquinazolin-4-amines as potent and selective inhibitors of cdc2-like kinases (Clk)

(2009) Bryan T. Mott et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and evaluation of fused bispyrimidinoacridines as novel pentacyclic analogues of quadruplex-binder BRACO-19

(2009) Julien Debray et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A rapid and versatile synthesis of novel pyrimido[5,4-b]carbazoles

(2009) Anna Caruso et al.   TETRAHEDRON

Concise Synthesis of 2-Amino-4(3H)-quinazolinones from Simple (Hetero)aromatic Amines

(2008) Walid Zeghida et al.   JOURNAL OF ORGANIC CHEMISTRY

Quinoline, quinazoline and acridonealkaloids

(2007) Joseph P. Michael   NATURAL PRODUCT REPORTS