β-Keto sulfones: preparation and application in organic synthesis

Multicomponent Reactions of β-Ketosulfones and Formaldehyde in a Bio-Based Binary Mixture Solvent System Composed of Meglumine and Gluconic Acid Aqueous Solution

(2012) Jie Yang et al.   ADVANCED SYNTHESIS & CATALYSIS

Design, synthesis and biological evaluation of novel (E)-α-benzylsulfonyl chalcone derivatives as potential BRAF inhibitors

(2012) Qing-Shan Li et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthesis of Isoxazole Triflones

(2012) Hiroyuki Kawai et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Ionic Liquid-Supported Sulfonyl Azide and Its Application in Diazotransfer Reaction

(2012) Manoj Kumar Muthyala et al.   JOURNAL OF ORGANIC CHEMISTRY

Three-Component Reaction ofβ-Ketosulfone, Formaldehyde, and Thiol or Thiophenol in Water

(2012) Yuying Du et al.   PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS

A Regioselective Catalyst- and Additive-Free Synthesis of β-Keto Sulfones from Aryl Acetylenes and Sodium Arenesulfinates

(2012) Bojja Sreedhar et al.   SYNLETT

Synthesis of α-Diazo Carbonyl Compounds with the Shelf-Stable Diazo Transfer Reagent Nonafluorobutanesulfonyl Azide

(2011) Jose Luis Chiara et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of 3-substituted 1,5-aldehyde estersvia an organocatalytic highly enantioselective conjugate addition of new carbonylmethyl 2-pyridinylsulfone to enals

(2011) Jing Deng et al.   CHEMICAL COMMUNICATIONS

Synthesis and chemical properties of cyclic β-keto sulfones (review)

(2011) O. O. Shyshkina et al.   Chemistry of Heterocyclic Compounds

Single step synthesis of new fused pyrimidine derivatives and their evaluation as potent Aurora-A kinase inhibitors

(2011) Mohamed R. Shaaban et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Dual Secondary Amine/N-Heterocyclic Carbene Catalysis in the Asymmetric Michael/Cross-Benzoin Cascade Reaction of β-Oxo Sulfones with Enals

(2011) Dieter Enders et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Practical Synthesis of β-Acyl and β-Alkoxycarbonyl Heterocyclic Sulfones

(2011) Jiří Pospíšil et al.   JOURNAL OF ORGANIC CHEMISTRY

β-(Trifluoromethyl)vinyl Sulfonium Salts: Preparation and Reactions with Active Methylene and Methenyl Compounds

(2011) Hao Lin et al.   JOURNAL OF ORGANIC CHEMISTRY

Rhenium-Catalyzed Regio- and Stereoselective Addition of Two Carbon Units to Terminal Alkynes via Carbon–Carbon Bond Cleavage of β-Keto Sulfones

(2011) Yoichiro Kuninobu et al.   ORGANIC LETTERS

Diaminomethylidene derivatives of β-oxo sulfones as potential reagents in heterocyclic synthesis and chelating ligands

(2011) V. A. Voronkova et al.   RUSSIAN CHEMICAL BULLETIN

Zinc-Mediated Tandem-One-Pot Facile Synthesis of 1-(Arylsulfonyl) Aryl/Heteryl Methanes: A Case of C‒S Bond Formation

(2011) K. Srinivas et al.   SYNTHETIC COMMUNICATIONS

Simple Strategy for Sulfonyl Ethynylogs of Coumarins

(2011) Nalajam Guravaiah et al.   SYNTHETIC COMMUNICATIONS

Unexpected formation of fluorine-containing tetrahydrocarbazole during the reaction of indole, paraformaldehyde, and fluorine-containing β-ketoesters

(2011) Wan Pang et al.   TETRAHEDRON

Ethyl-2-(2-chloroethyl)acrylate: a new very versatile α-cyclopropylester cation synthon. Efficient synthesis of cyclopropane ester derivatives by Michael addition-induced cyclization reaction

(2011) Mathilde Lachia et al.   TETRAHEDRON LETTERS

Stereoselective synthesis of ambiphilic alkenes via regioselective methylation of α-trifluoromethanesulfonyl carbonyl compounds with trimethylsilyldiazomethane

(2011) Han Il Kong et al.   TETRAHEDRON LETTERS

1-Butyl-3-methylimidazolium p-toluenesulfinate: a novel reagent for synthesis of sulfones and β-ketosulfones in ionic liquid

(2011) Anil Kumar et al.   TETRAHEDRON LETTERS

Amine-catalyzed (3+n) annulations of 2-(acetoxymethyl)buta-2,3-dienoates with 1,n-bisnucleophiles (n = 3–5)

(2010) Chaolong Li et al.   CHEMICAL COMMUNICATIONS

Synthesis of Chiral Cyclic Nitrones by Asymmetric Addition of β-Ketosulfones to Nitroalkenes followed by Reductive Cyclization

(2010) Olga García Mancheño et al.   CHEMISTRY-A EUROPEAN JOURNAL

Catalytic Asymmetric Michael Reactions of α,β-Unsaturated Ketones with Sulfonyl-Containing Nucleophiles: Chiral Synthesis of (R)-Muscone and (S)-Celery Ketone

(2010) Xiaomin Sun et al.   CHEMISTRY-A EUROPEAN JOURNAL

p-Toluenesulfonic Acid Promoted Annulation of 2-Alkynylanilines with Activated Ketones: Efficient Synthesis of 4-Alkyl-2,3-Disubstituted Quinolines

(2010) Changlan Peng et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Highly Enantioselective Intramolecular Copper Catalyzed C−H Insertion Reactions of α-Diazosulfones

(2010) Christopher J. Flynn et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium(I)-Catalyzed Addition of Arylboronic Acids to (Benzyl-/Arylsulfonyl)acetonitriles: Efficient Synthesis of (Z)-β-Sulfonylvinylamines and β-Keto Sulfones

(2010) Gavin Chit Tsui et al.   ORGANIC LETTERS

A Facile Access to Some New Pyrazole, 1,3,4-Thiadiazole, and Thiophene Derivatives via β-Ketosulfones

(2010) Kamal Dawood et al.   PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS

Synthesis of a New Class of Sulfone-Linked 3-([1,2,3]-Thiadazol-4-yl)-chromen-2-ones

(2010) Nalajam Guravaiah et al.   PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS

New approach to 5-arylsulfonyl-substituted 1,2-dihydropyrimidin-2-ones via base-induced chloroform elimination from 4-trichloromethyl-1,2,3,4-tetrahydropyrimidin-2-ones

(2010) Anastasia A. Fesenko et al.   TETRAHEDRON

Enantioselective reduction of α-substituted ketones mediated by the boronate ester TarB-NO2

(2010) Scott Eagon et al.   TETRAHEDRON LETTERS

Reaction of 6-aryl- or styryl-4-methylsulfanyl-2-oxo-2H-pyrans with active methylene compounds and fluorescence properties of the products

(2009) Naoko Mizuyama et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

4H-1-Benzopyrans by a tandem SN2-SNAr reaction

(2009) Richard A. Bunce et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

A Benzannulation Protocol To Prepare Substituted Aryl Amines Using a Michael-Aldol Reaction of β-Keto Sulfones

(2009) Sezgin Kiren et al.   JOURNAL OF ORGANIC CHEMISTRY

Rhodium Carbene Routes to Oxazoles and Thiazoles. Catalyst Effects in the Synthesis of Oxazole and Thiazole Carboxylates, Phosphonates, and Sulfones

(2009) Baolu Shi et al.   JOURNAL OF ORGANIC CHEMISTRY

(Arylsulfonyl)acetones and -acetonitriles: New Activated Methylenic Building Blocks for Synthesis of 1,2,3-Triazoles

(2009) Nazariy Pokhodylo et al.   SYNTHESIS-STUTTGART

A Mitsunobu route to C-glycosides

(2009) Paolo Pasetto et al.   TETRAHEDRON

Ring expansion reaction of α-sulfonyl cyclic ketones via insertion of arynes into C–C: a facile and mild access to medium- and large-sized benzannulated carbocycles

(2009) Tiexin Zhang et al.   TETRAHEDRON LETTERS

Facile polyethylene glycol (PEG-400) promoted synthesis of some new heteryl (E)-styryl sulfones

(2009) Nalajam Guravaiah et al.   JOURNAL OF CHEMICAL RESEARCH

Solvent-free synthesis of new heteryl β-ketosulfones

(2009) Nalajam Guravaiah et al.   JOURNAL OF CHEMICAL RESEARCH

Synthesis and analgesic/anti-inflammatory evaluation of fused heterocyclic ring systems incorporating phenylsulfonyl moiety

(2008) Mohamed R. Shaaban et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Dynamic kinetic resolution of β-keto sulfonesvia asymmetric transfer hydrogenation

(2008) Zhenhua Ding et al.   CHEMICAL COMMUNICATIONS

Synthesis of stable arsonium and sulfur ylides from perfluoroalkanesulfonyl diazocarbonyl compounds and their X-ray diffraction analysis

(2008) Wan Pang et al.   JOURNAL OF FLUORINE CHEMISTRY

Copper(II)−Bis(oxazoline) Catalyzed Asymmetric Diels−Alder Reaction with α′-Arylsulfonyl Enones as Dienophiles

(2008) Santiago Barroso et al.   JOURNAL OF ORGANIC CHEMISTRY

A Versatile and Highly Stereoselective Access to Vinyl Triflates Derived from 1,3-Dicarbonyl and Related Compounds

(2008) Simon Specklin et al.   JOURNAL OF ORGANIC CHEMISTRY

Studies on the Chemistry and Reactivity of α-Substituted Ketones in Isonitrile-Based Multicomponent Reactions†

(2008) Lijun Fan et al.   JOURNAL OF ORGANIC CHEMISTRY

A Novel and Convenient Protocol for Synthesis of Pyridazines

(2008) Orazio A. Attanasi et al.   ORGANIC LETTERS

Multicomponent Reactions as a Powerful Tool for Generic Drug Synthesis

(2008) Cédric Kalinski et al.   SYNTHESIS-STUTTGART

Application of HOF·CH3CN to the synthesis of glycosyl sulfones

(2008) Goreti Ribeiro Morais et al.   TETRAHEDRON

α-Fluorination of β-ketosulfones by Selectfluor™ F–TEDA–BF4

(2008) Hossein Loghmani-Khouzani et al.   TETRAHEDRON

Microwave-assisted manganese(III) acetate based oxidative cyclizations of alkenes with β-ketosulfones

(2008) Christophe Curti et al.   TETRAHEDRON

Regioselective synthesis of 1,2,4,5-tetrasubstituted pyridines from Baylis–Hillman adducts via consecutive [3+2+1] annulation protocol

(2008) Sung Hwan Kim et al.   TETRAHEDRON LETTERS

Synthesis of enantiomerically enriched secondary and tertiary phenylthio- and phenoxy-aldols

(2008) Angela M. Bernard et al.   TETRAHEDRON LETTERS

First synthesis of 4-(arylsulfonyl)phenols by regioselective [3+3] cyclocondensations of 1,3-bis(silyloxy)-1,3-butadienes with 2-arylsulfonyl-3-ethoxy-2-en-1-ones

(2008) Abdolmajid Riahi et al.   TETRAHEDRON LETTERS