SYMPOSIUM REVIEW: Revealing the structural basis of action of hERG potassium channel activators and blockers
出版年份 2010 全文链接
标题
SYMPOSIUM REVIEW: Revealing the structural basis of action of hERG potassium channel activators and blockers
作者
关键词
-
出版物
JOURNAL OF PHYSIOLOGY-LONDON
Volume 588, Issue 17, Pages 3157-3167
出版商
Wiley
发表日期
2010-07-20
DOI
10.1113/jphysiol.2010.194670
参考文献
相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。- The amiodarone derivative KB130015 activates hERG1 potassium channels via a novel mechanism
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- Electrophysiologic characterization of a novel hERG channel activator
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- Docking Model of Drug Binding to the Human Ether-à-go-go Potassium Channel Guided by Tandem Dimer Mutant Patch-Clamp Data: A Synergic Approach
- (2009) Yumi N. Imai et al. JOURNAL OF MEDICINAL CHEMISTRY
- Pharmacological Removal of Human Ether-a-go-go-Related Gene Potassium Channel Inactivation by 3-Nitro-N-(4-phenoxyphenyl) Benzamide (ICA-105574)
- (2009) A. C. Gerlach et al. MOLECULAR PHARMACOLOGY
- PD-118057 contacts the pore helix of hERG1 channels to attenuate inactivation and enhance K+ conductance
- (2009) M. Perry et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- hERG1 channel activators: A new anti-arrhythmic principle
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- Insight into the Mechanism of Inactivation and pH Sensitivity in Potassium Channels from Molecular Dynamics Simulations†
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- Pharmacology of the short QT syndrome N588K-hERG K+channel mutation: differential impact on selected class I and class III antiarrhythmic drugs
- (2008) M J McPate et al. BRITISH JOURNAL OF PHARMACOLOGY
- The Pore Domain Outer Helix Contributes to Both Activation and Inactivation of the hERG K+Channel
- (2008) Pengchu Ju et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Molecular Determinants of hERG Channel Block by Terfenadine and Cisapride
- (2008) Kaichiro Kamiya et al. JOURNAL OF PHARMACOLOGICAL SCIENCES
- Topological Mapping of the Asymmetric Drug Binding to the Human Ether-a-go-go-Related Gene Product (HERG) Potassium Channel by Use of Tandem Dimers
- (2008) T. Myokai et al. MOLECULAR PHARMACOLOGY
- Probing the Binding Sites and Mechanisms of Action of Two Human Ether-a-go-go-Related Gene Channel Activators, 1,3-bis-(2-Hydroxy-5-trifluoromethyl-phenyl)-urea (NS1643) and 2-[2-(3,4-Dichloro-phenyl)-2,3-dihydro-1H-isoindol-5-ylamino]-nicotinic acid (PD307243)
- (2008) X. Xu et al. MOLECULAR PHARMACOLOGY
- Drug Binding to the Inactivated State Is Necessary but Not Sufficient for High-Affinity Binding to Human Ether-a-go-go-Related Gene Channels
- (2008) M. J. Perrin et al. MOLECULAR PHARMACOLOGY
- The hERG potassium channel and hERG screening for drug-induced torsades de pointes
- (2008) Jules C. Hancox et al. PHARMACOLOGY & THERAPEUTICS
- State dependent dissociation of HERG channel inhibitors
- (2007) D Stork et al. BRITISH JOURNAL OF PHARMACOLOGY
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