期刊
JOURNAL OF ORGANIC CHEMISTRY
卷 78, 期 23, 页码 12144-12153出版社
AMER CHEMICAL SOC
DOI: 10.1021/jo402132p
关键词
-
资金
- National Institutes of Health [GM-64444]
- Ministry of Education of the Perm Krai
Bronsted acid-catalyzed one-pot synthesis of indoles from o-aminobenzyl alcohols and furans has been developed. This method operates via the in situ formation of aminobenzylfuran, followed by its recyclization into the indole core. The method proved to be efficient for substrates possessing different functional groups, including -OMe, -CO2Cy, and -Br. The resulting indoles can easily be transformed into diverse scaffolds, including 2,3- and 1,2-fused indoles, and indoles possessing an alpha,beta-unsaturated ketone moiety at the C-2 position.
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