Discovery and Characterization of 6-{4-[3-(R)-2-Methylpyrrolidin-1-yl)propoxy]phenyl}-2H-pyridazin-3-one (CEP-26401, Irdabisant): A Potent, Selective Histamine H3Receptor Inverse Agonist

标题
Discovery and Characterization of 6-{4-[3-(R)-2-Methylpyrrolidin-1-yl)propoxy]phenyl}-2H-pyridazin-3-one (CEP-26401, Irdabisant): A Potent, Selective Histamine H3Receptor Inverse Agonist
作者
关键词
-
出版物
JOURNAL OF MEDICINAL CHEMISTRY
Volume 54, Issue 13, Pages 4781-4792
出版商
American Chemical Society (ACS)
发表日期
2011-06-03
DOI
10.1021/jm200401v

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