期刊
ORGANIC LETTERS
卷 17, 期 23, 页码 5906-5909出版社
AMER CHEMICAL SOC
DOI: 10.1021/acs.orglett.5b03104
关键词
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资金
- Research Grants Council of Hong Kong [CRF: C5023-14G]
- General Research Fund [PolyU 153008/14P]
- State Key Laboratory of Chirosciences
The first general palladium catalyst for the phosphorylation of aryl mesylates and tosylates is reported. The newly developed system exhibits excellent functional group compatibility. For instance, free amino, keto, ester, and amido groups, as well as heterocycles, remain intact during the course of reaction. The mesylated derivatives of biologically active compounds such as 17 beta-estradiol and 6-hydroxyflavone are also shown to be applicable substrates. A one-pot phosphorylation-amination sequence is described for the facile synthesis of potential phannacophores.
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