Synthesis of BODIPY Derivatives Substituted with Various Bioconjugatable Linker Groups: A Construction Kit for Fluorescent Labeling of Receptor Ligands

Novel fluorescent antagonist as a molecular probe in A3 adenosine receptor binding assays using flow cytometry

(2012) Eszter Kozma et al.   BIOCHEMICAL PHARMACOLOGY

Synthesis and structure–activity relationships of 2-hydrazinyladenosine derivatives as A2A adenosine receptor ligands

(2012) Ali El-Tayeb et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Fragment Screening at Adenosine-A3 Receptors in Living Cells Using a Fluorescence-Based Binding Assay

(2012) Leigh A. Stoddart et al.   CHEMISTRY & BIOLOGY

Water-Soluble Red-Emitting Distyryl-Borondipyrromethene (BODIPY) Dyes for Biolabeling

(2012) Song-lin Niu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Fluorescent Derivatives of AC-42 To Probe Bitopic Orthosteric/Allosteric Binding Mechanisms on Muscarinic M1 Receptors

(2012) Sandrine B. Daval et al.   JOURNAL OF MEDICINAL CHEMISTRY

Highly Potent and Selective Fluorescent Antagonists of the Human Adenosine A3 Receptor Based on the 1,2,4-Triazolo[4,3-a]quinoxalin-1-one Scaffold

(2012) Andrea J. Vernall et al.   JOURNAL OF MEDICINAL CHEMISTRY

Oxidative Coupling of 1,7,8-Unsubstituted BODIPYs: Synthesis and Electrochemical and Spectroscopic Properties

(2012) Arnaud Poirel et al.   JOURNAL OF ORGANIC CHEMISTRY

8-AminoBODIPYs: Cyanines or Hemicyanines? The Effect of the Coplanarity of the Amino Group on Their Optical Properties

(2012) Carlos A. Osorio-Martínez et al.   JOURNAL OF ORGANIC CHEMISTRY

A General Synthetic Route to 3,5-Substituted Boron Dipyrromethenes: Applications and Properties

(2012) Gilles Ulrich et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and photodynamic activity of a panel of BODIPY dyes

(2012) Stefano Banfi et al.   JOURNAL OF PHOTOCHEMISTRY AND PHOTOBIOLOGY B-BIOLOGY

The four cysteine residues in the second extracellular loop of the human adenosine A2B receptor: Role in ligand binding and receptor function

(2011) Anke C. Schiedel et al.   BIOCHEMICAL PHARMACOLOGY

GPCR Ligand Dendrimer (GLiDe) Conjugates: Adenosine Receptor Interactions of a Series of Multivalent Xanthine Antagonists

(2011) Angela Kecskés et al.   BIOCONJUGATE CHEMISTRY

A BODIPY-Cyclooctyne for Protein Imaging in Live Cells

(2011) Kimberly E. Beatty et al.   CHEMBIOCHEM

Fluorescent indicators based on BODIPY

(2011) Noël Boens et al.   CHEMICAL SOCIETY REVIEWS

Advances in the chemistry of small molecule fluorescent probes

(2011) Laura M Wysocki et al.   CURRENT OPINION IN CHEMICAL BIOLOGY

Some observations relating to the stability of the BODIPY fluorophore under acidic and basic conditions

(2011) Lijing Yang et al.   DYES AND PIGMENTS

Synthesis and Characterization of High-Affinity 4,4-Difluoro-4-bora-3a,4a-diaza-s-indacene-Labeled Fluorescent Ligands for Human β-Adrenoceptors

(2011) Jillian G. Baker et al.   JOURNAL OF MEDICINAL CHEMISTRY

Highly Substituted Bodipy Dyes with Spectroscopic Features Sensitive to the Environment

(2011) Thomas Bura et al.   JOURNAL OF ORGANIC CHEMISTRY

Red-Emission Fluorescent Probe Sensing Cadmium and Pyrophosphate Selectively in Aqueous Solution

(2011) Tanyu Cheng et al.   ORGANIC LETTERS

New potent, short-linker BODIPY-630/650™ labelled fluorescent adenosine receptor agonists

(2011) Clare L. Dale et al.   MedChemComm

Development of Polar Adenosine A2A Receptor Agonists for Inflammatory Bowel Disease: Synergism with A2B Antagonists

(2011) Ali El-Tayeb et al.   ACS Medicinal Chemistry Letters

Novel Alexa Fluor-488 labeled antagonist of the A2A adenosine receptor: Application to a fluorescence polarization-based receptor binding assay

(2010) Miklós Kecskés et al.   BIOCHEMICAL PHARMACOLOGY

Recent developments in adenosine receptor ligands and their potential as novel drugs

(2010) Christa E. Müller et al.   BIOCHIMICA ET BIOPHYSICA ACTA-BIOMEMBRANES

Polyamidoamine (PAMAM) Dendrimer Conjugates of “Clickable” Agonists of the A3Adenosine Receptor and Coactivation of the P2Y14Receptor by a Tethered Nucleotide

(2010) Dilip K. Tosh et al.   BIOCONJUGATE CHEMISTRY

Molecular probes for the A2A adenosine receptor based on a pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine scaffold

(2010) T. Santhosh Kumar et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Influence of fluorophore and linker composition on the pharmacology of fluorescent adenosine A1 receptor ligands

(2010) Jillian G Baker et al.   BRITISH JOURNAL OF PHARMACOLOGY

“Alive” dyes as fluorescent sensors: fluorophore, mechanism, receptor and images in living cells

(2010) Xuhong Qian et al.   CHEMICAL COMMUNICATIONS

Antagonist Selective Modulation of Adenosine A1 and A3 Receptor Pharmacology by the Food Dye Brilliant Black BN: Evidence for Allosteric Interactions

(2010) L. T. May et al.   MOLECULAR PHARMACOLOGY

2-Dialkynyl derivatives of (N)-methanocarba nucleosides: ‘Clickable’ A3 adenosine receptor-selective agonists

(2009) Dilip K. Tosh et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, spectroscopic properties and protein labeling of water soluble 3,5-disubstituted boron dipyrromethenes

(2009) Özlem Dilek et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Solid-State Gas Sensors Developed from Functional Difluoroboradiazaindacene Dyes

(2009) Raymond Ziessel et al.   CHEMISTRY-A EUROPEAN JOURNAL

1-Alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: Development and Characterization of Adenosine A2BReceptor Antagonists and a New Radioligand with Subnanomolar Affinity and Subtype Specificity

(2009) Thomas Borrmann et al.   JOURNAL OF MEDICINAL CHEMISTRY

Nucleoside-5′-monophosphates as Prodrugs of Adenosine A2AReceptor Agonists Activated by ecto-5′-Nucleotidase†† Contribution to celebrate the 100th anniversary of the Division of Medicinal Chemistry of the American Chemical Society.

(2009) Ali El-Tayeb et al.   JOURNAL OF MEDICINAL CHEMISTRY

Carboxyl BODIPY Dyes from Bicarboxylic Anhydrides: One-Pot Preparation, Spectral Properties, Photostability, and Biolabeling

(2009) Dongchuan Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

A highly selective and sensitive fluorescent turn-on sensor for Hg2+ and its application in live cell imaging

(2009) Hua Lu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Water-Soluble BODIPY Derivatives

(2009) Song Lin Niu et al.   ORGANIC LETTERS

Fluorescent DNA Base Modifications and Substitutes: Multiple Fluorophore Labeling and the DETEQ Concept

(2008) Hans-Achim Wagenknecht   Annals of the New York Academy of Sciences

Fluorescent GPCR Ligands as New Tools in Pharmacology

(2008) Kamil Kuder et al.   CURRENT MEDICINAL CHEMISTRY

Adenosine A2A receptor dynamics studied with the novel fluorescent agonist Alexa488-APEC

(2008) Frank Brand et al.   EUROPEAN JOURNAL OF PHARMACOLOGY

The Chemistry of Fluorescent Bodipy Dyes: Versatility Unsurpassed

(2007) Gilles Ulrich et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Agonist-occupied A3 adenosine receptors exist within heterogeneous complexes in membrane microdomains of individual living cells

(2007) Y. Cordeaux et al.   FASEB JOURNAL