Structure-based Virtual Screening and Identification of a Novel Androgen Receptor Antagonist

Mechanism of Androgen Receptor Antagonism by Bicalutamide in the Treatment of Prostate Cancer

(2011) D. J. Osguthorpe et al.   BIOCHEMISTRY

Inhibitors of Androgen Receptor Activation Function-2 (AF2) Site Identified through Virtual Screening

(2011) Peter Axerio-Cilies et al.   JOURNAL OF MEDICINAL CHEMISTRY

Regression of Castrate-Recurrent Prostate Cancer by a Small-Molecule Inhibitor of the Amino-Terminus Domain of the Androgen Receptor

(2010) Raymond J. Andersen et al.   CANCER CELL

Resveratrol regulates the PTEN/AKT pathway through androgen receptor-dependent and -independent mechanisms in prostate cancer cell lines

(2010) Yu Wang et al.   HUMAN MOLECULAR GENETICS

Structure−Activity Relationship for Thiohydantoin Androgen Receptor Antagonists for Castration-Resistant Prostate Cancer (CRPC)

(2010) Michael E. Jung et al.   JOURNAL OF MEDICINAL CHEMISTRY

Limitations of MTT and MTS-Based Assays for Measurement of Antiproliferative Activity of Green Tea Polyphenols

(2010) Piwen Wang et al.   PLoS One

Androgen Receptor Regulates a Distinct Transcription Program in Androgen-Independent Prostate Cancer

(2009) Qianben Wang et al.   CELL

Nonsteroidal Selective Androgen Receptor Modulators (SARMs): Dissociating the Anabolic and Androgenic Activities of the Androgen Receptor for Therapeutic Benefit

(2009) Michael L. Mohler et al.   JOURNAL OF MEDICINAL CHEMISTRY

HDAC6 Regulates Androgen Receptor Hypersensitivity and Nuclear Localization via Modulating Hsp90 Acetylation in Castration-Resistant Prostate Cancer

(2009) Junkui Ai et al.   MOLECULAR ENDOCRINOLOGY

Development of a Second-Generation Antiandrogen for Treatment of Advanced Prostate Cancer

(2009) C. Tran et al.   SCIENCE

Hepatocyte nuclear factor-3 alpha (HNF-3α) negatively regulates androgen receptor transactivation in prostate cancer cells

(2008) Hyun Joo Lee et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS

Cancer Statistics, 2008

(2008) A. Jemal et al.   CA-A CANCER JOURNAL FOR CLINICIANS

Computationally Identified Novel Diphenyl- and Phenylpyridine Androgen Receptor Antagonist Structures

(2008) Annu A. Söderholm et al.   Journal of Chemical Information and Modeling

Reduced testicular steroidogenesis in tumor necrosis factor-α knockout mice

(2008) Ji Ho Suh et al.   JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY

Regulation of androgen receptor transcriptional activity by rapamycin in prostate cancer cell proliferation and survival

(2008) Y Wang et al.   ONCOGENE

CR6-Interacting Factor 1 Represses the Transactivation of Androgen Receptor by Direct Interaction

(2007) Ji Ho Suh et al.   MOLECULAR ENDOCRINOLOGY