G Protein-Coupled Receptor Signaling Analysis Using Homogenous Time-Resolved Förster Resonance Energy Transfer (HTRF®) Technology

Signalling bias in new drug discovery: detection, quantification and therapeutic impact

(2013) Terry Kenakin et al.   NATURE REVIEWS DRUG DISCOVERY

Novel Strategies in Drug Discovery of the Calcium-Sensing Receptor Based on Biased Signaling

(2012) Alex Rojas Bie Thomsen et al.   CURRENT DRUG TARGETS

An update of novel screening methods for GPCR in drug discovery

(2012) Linjie Chen et al.   Expert Opinion on Drug Discovery

Using label-free screening technology to improve efficiency in drug discovery

(2012) Reena Halai et al.   Expert Opinion on Drug Discovery

Biased agonism of the calcium-sensing receptor

(2011) Alex Rojas Bie Thomsen et al.   CELL CALCIUM

Monitoring Gq-coupled receptor response through inositol phosphate quantification with the IP-One assay

(2011) Eric Trinquet et al.   Expert Opinion on Drug Discovery

The development of label-free cellular assays for drug discovery

(2011) Ye Fang   Expert Opinion on Drug Discovery

Elusive equilibrium: the challenge of interpreting receptor pharmacology using calcium assays

(2010) Steven J Charlton et al.   BRITISH JOURNAL OF PHARMACOLOGY

Functional Selectivity and Biased Receptor Signaling

(2010) T. Kenakin   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

Deconvolution of complex G protein–coupled receptor signaling in live cells using dynamic mass redistribution measurements

(2010) Ralf Schröder et al.   NATURE BIOTECHNOLOGY

Time-resolved luminescence resonance energy transfer imaging of protein-protein interactions in living cells

(2010) H. E. Rajapakse et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Development of a homogeneous competitive immunoassay for phosphorylated protein antigen based on the enhanced fluorescence resonance energy transfer technology

(2009) Yoshiyuki Ohiro et al.   JOURNAL OF BIOSCIENCE AND BIOENGINEERING

A One-Day, Dispense-Only IP-One HTRF Assay for High-Throughput Screening of Gαq Protein-Coupled Receptors: Towards Cells as Reagents

(2008) Christian Bergsdorf et al.   ASSAY AND DRUG DEVELOPMENT TECHNOLOGIES

Current status of HTRF®technology in kinase assays

(2008) Yong Jia   Expert Opinion on Drug Discovery