The Synthesis and Glycoside Formation of Polyfluorinated Carbohydrates

Fluorinated Nucleosides: Synthesis, Modulation in Conformation and Therapeutic Application

(2022) Shantanu Pal et al.   CHEMICAL RECORD

Development of α-Selective Glycosylation for the Synthesis of Deoxyfluorinated TN Antigen Analogues

(2021) Martin Kurfiřt et al.   JOURNAL OF ORGANIC CHEMISTRY

Polyfluoroglycoside Synthesis via Simple Alkylation of an Anomeric Hydroxyl Group: Access to Fluoroetoposide Analogues

(2021) Thomas Tremblay et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of multiply fluorinated N-acetyl-D-glucosamine and D-galactosamine analogs via the corresponding deoxyfluorinated glucosazide and galactosazide phenyl thioglycosides

(2021) Vojtěch Hamala et al.   Beilstein Journal of Organic Chemistry

Anti-glycan antibodies: roles in human disease

(2021) J. Sebastian Temme et al.   BIOCHEMICAL JOURNAL

Recent advances on smart glycoconjugate vaccines in infections and cancer

(2021) Marko Anderluh et al.   FEBS Journal

Carbohydrate-Based Macromolecular Biomaterials

(2021) Lu Su et al.   CHEMICAL REVIEWS

Selectively Deoxyfluorinated N ‐Acetyllactosamine Analogues as 19 F NMR Probes to Study Carbohydrate‐Galectin Interactions

(2021) Martin Kurfiřt et al.   CHEMISTRY-A EUROPEAN JOURNAL

Electrochemical Trifluoromethylation of Glycals

(2021) Miao Liu et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Structural Characteristics of all Mono- and Difluorinated 4,6-Dideoxy-d-xylo-hexopyranoses

(2021) David E. Wheatley et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of fluorinated thiodigalactoside analogues

(2021) Jacob St-Gelais et al.   CARBOHYDRATE RESEARCH

Sweetening Pharmaceutical Radiochemistry by 18F-Fluoroglycosylation: Recent Progress and Future Prospects

(2021) Sandip S. Shinde et al.   Pharmaceuticals

Conformational studies of oligosaccharides

(2020) Yang Yu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Galactofuranose-Related Enzymes: Challenges and Hopes

(2020) Mateja Seničar et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

Addressing the structural complexity of fluorinated glucose analogues: Insight into lipophilicities and solvation effects

(2020) Jacob St-Gelais et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthetic Fluorinated l-Fucose Analogs Inhibit Proliferation of Cancer Cells and Primary Endothelial Cells

(2020) Yuanwei Dai et al.   ACS Chemical Biology

The role of fluorine in glycomimetic drug design

(2020) Rachel Hevey   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis and Anti-HCV Activity of Sugar-Modified Guanosine Analogues: Discovery of AL-611 as an HCV NS5B Polymerase Inhibitor for the Treatment of Chronic Hepatitis C

(2020) Guangyi Wang et al.   JOURNAL OF MEDICINAL CHEMISTRY

Fluorine effect in nucleophilic fluorination at C4 of 1,6-anhydro-2,3-dideoxy-2,3-difluoro-β-D-hexopyranose

(2020) Danny Lainé et al.   Beilstein Journal of Organic Chemistry

From Carbohydrates to Complex Organofluorines: Synthesis, Conformation, and Lipophilicity of Multivicinal‐Fluorine‐Containing Hexitol Analogues

(2020) Danny Lainé et al.   CHEMISTRY-A EUROPEAN JOURNAL

Fluorinated Carbohydrates as Lectin Ligands: Simultaneous Screening of a Monosaccharide Library and Chemical Mapping by 19F NMR Spectroscopy

(2020) J. Daniel Martínez et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Conformational Analysis of Fluorinated Uridine Analogues Provide Insight into a Neighbouring-Group Participation Mechanism

(2020) Freideriki Michailidou et al.   MOLECULES

Virus recognition of glycan receptors

(2019) Andrew J Thompson et al.   Current Opinion in Virology

Synthesis of 2-fluoro-substituted and 2,6-modified purine 2′,3′-dideoxy-2′,3′-difluoro-d-arabinofuranosyl nucleosides from d-xylose

(2019) Grigorii G. Sivets et al.   TETRAHEDRON

Regio- and Chemoselective Deprotection of Primary Acetates by Zirconium Hydrides

(2019) Marine Gavel et al.   ORGANIC LETTERS

Oligosaccharide Synthesis and Translational Innovation

(2019) Larissa Krasnova et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Hydrogen Bonding Phase-Transfer Catalysis with Potassium Fluoride: Enantioselective Synthesis of β-Fluoroamines

(2019) Gabriele Pupo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of 2,3,4-Trideoxy-2,3,4-trifluoroglucose

(2019) Lucas Quiquempoix et al.   JOURNAL OF ORGANIC CHEMISTRY

Nuclear Imaging of Glucose Metabolism: Beyond 18F-FDG

(2019) Han Feng et al.   Contrast Media & Molecular Imaging

Stereospecific α-Sialylation by Site-Selective Fluorination

(2019) Taiki Hayashi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Exploitation of glycosylation in enveloped virus pathobiology

(2019) Yasunori Watanabe et al.   BIOCHIMICA ET BIOPHYSICA ACTA-GENERAL SUBJECTS

Stereoselective Synthesis of Fluorinated Galactopyranosides as Potential Molecular Probes for Galactophilic Proteins: Assessment of Monofluorogalactoside–LecA Interactions

(2019) Vincent Denavit et al.   CHEMISTRY-A EUROPEAN JOURNAL

Exploring the chemistry of non‐sticky sugars: Synthesis of polyfluorinated carbohydrate analogs of D‐allopyranose

(2019) Vincent Denavit et al.   CHEMISTRY-A EUROPEAN JOURNAL

9-Azido-9-deoxy-2,3-difluorosialic Acid as a Subnanomolar Inhibitor against Bacterial Sialidases

(2019) Wanqing Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Stereoselectivity in Glycosylation with Deoxofluorinated Glucosazide and Galactosazide Thiodonors

(2019) Martin Kurfiřt et al.   JOURNAL OF ORGANIC CHEMISTRY

Targeting the Chondroitin Sulfate Proteoglycans: Evaluating Fluorinated Glucosamines and Xylosides in Screens Pertinent to Multiple Sclerosis

(2019) Erin L. Stephenson et al.   ACS Central Science

Structural and Computational Analysis of 2-Halogeno-Glycosyl Cations in Superacid: An extansive Platform

(2019) Ludivine Lebedel et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and Lipophilicity of Trifluorinated Analogues of Glucose

(2019) Jacob St-Gelais et al.   JOURNAL OF ORGANIC CHEMISTRY

Design and synthesis of glycomimetics: Recent advances

(2019) Alice Tamburrini et al.   MEDICINAL RESEARCH REVIEWS

Structural Studies Using Unnatural Oligosaccharides: Toward Sugar Foldamers

(2019) Theodore Tyrikos-Ergas et al.   BIOMACROMOLECULES

XtalFluor-E: A useful and versatile reagent in organic transformations

(2019) Leyla Mohammadkhani et al.   JOURNAL OF FLUORINE CHEMISTRY

Novel NMR Avenues to Explore the Conformation and Interactions of Glycans

(2019) Pablo Valverde et al.   ACS Omega

Design, properties and applications of fluorinated and fluoroalkylated N-containing monosaccharides and their analogues

(2019) Monika Bilska-Markowska et al.   JOURNAL OF FLUORINE CHEMISTRY

Open-Shell Fluorination of Alkyl Bromides: Unexpected Selectivity in a Silyl Radical-Mediated Chain Process

(2019) Gabrielle H. Lovett et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The recognition of glycans by protein receptors. Insights from NMR spectroscopy

(2018) Ana Ardá et al.   CHEMICAL COMMUNICATIONS

Applications of controlled inversion strategies in carbohydrate synthesis

(2018) Wuqiong Song et al.   CHINESE CHEMICAL LETTERS

Synthesis of Fluorinated Leishmania Cap Trisaccharides for Diagnostic Tool and Vaccine Development

(2018) Andreas Baumann et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Double-Modified Xyloside Analogues for Probing the β4GalT7 Active Site

(2018) Daniel Willén et al.   JOURNAL OF ORGANIC CHEMISTRY

Deoxyfluorination with Sulfonyl Fluorides: Navigating Reaction Space with Machine Learning

(2018) Matthew K. Nielsen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Carbohydrate-based vaccines for oncotherapy

(2018) Meng-Man Wei et al.   MEDICINAL RESEARCH REVIEWS

Design, synthesis and biological evaluation of (2S,3R,4R,5S,6R)-5-fluoro-6-(hydroxymethyl)-2-aryltetrahydro-2H-pyran-3,4-diols as potent and orally active SGLT dual inhibitors

(2018) Guozhang Xu et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Re-Engineering Chemical Glycosylation: Direct, Metal-Free Anomeric O-Arylation of Unactivated Carbohydrates

(2018) Nicola Lucchetti et al.   CHEMISTRY-A EUROPEAN JOURNAL

Kinetics of Electrophilic Fluorinations of Enamines and Carbanions: Comparison of the Fluorinating Power of N–F Reagents

(2018) Daria S. Timofeeva et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A quantitative reactivity scale for electrophilic fluorinating reagents

(2018) Neshat Rozatian et al.   Chemical Science

Fluorinated Carbohydrates as Lectin Ligands: Synthesis of OH/F-Substituted N -Glycan Core Trimannoside and Epitope Mapping by 2D STD-TOCSYreF NMR spectroscopy

(2018) Tammo Diercks et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Domino Epoxide Ring-Opening Xanthate Migration Reaction: An Alternative Entry to Thiosugars

(2018) María B. Comba et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A Chiron approach towards the stereoselective synthesis of polyfluorinated carbohydrates

(2018) Vincent Denavit et al.   Nature Communications

Fluorinated nucleosides as an important class of anticancer and antiviral agents

(2017) Alessandra Cavaliere et al.   Future Medicinal Chemistry

Synthesis of Protected 3-Deoxy-3-fluoro- and 4-Deoxy-4-fluoro-d-galactopyranosides from Levoglucosan

(2017) Danny Lainé et al.   JOURNAL OF ORGANIC CHEMISTRY

Designer α1,6-Fucosidase Mutants Enable Direct Core Fucosylation of Intact N-Glycopeptides and N-Glycoproteins

(2017) Chao Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Recent Developments in the Deoxyfluorination of Alcohols and Phenols: New Reagents, Mechanistic Insights, and Applications

(2017) Xiang-Guo Hu et al.   SYNTHESIS-STUTTGART

Synthesis and antiviral evaluation of 2′,2′,3′,3′-tetrafluoro nucleoside analogs

(2017) Ozkan Sari et al.   TETRAHEDRON LETTERS

Synthesis and in vitro cytotoxicity of acetylated 3-fluoro, 4-fluoro and 3,4-difluoro analogs of D-glucosamine and D-galactosamine

(2016) Štěpán Horník et al.   Beilstein Journal of Organic Chemistry

Hydrogen-bond promoted nucleophilic fluorination: concept, mechanism and applications in positron emission tomography

(2016) Ji-Woong Lee et al.   CHEMICAL SOCIETY REVIEWS

Debenzylative Cycloetherification: An Overlooked Key Strategy for Complex Tetrahydrofuran Synthesis

(2016) Abdellatif Tikad et al.   CHEMISTRY-A EUROPEAN JOURNAL

Enantioselective Synthesis of Dideoxy-tetrafluorinated Hexoses

(2016) Samuel Golten et al.   JOURNAL OF ORGANIC CHEMISTRY

Hydrogen-Bonded Homoleptic Fluoride–Diarylurea Complexes: Structure, Reactivity, and Coordinating Power

(2016) Lukas Pfeifer et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Study of Uridine 5′-Diphosphate (UDP)-Galactopyranose Mutase Using UDP-5-Fluorogalactopyranose as a Probe: Incubation Results and Mechanistic Implications

(2016) Geng-Min Lin et al.   ORGANIC LETTERS

Structures of mammalian ER α-glucosidase II capture the binding modes of broad-spectrum iminosugar antivirals

(2016) Alessandro T. Caputo et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Synthesis of multivalent difluorinated zanamivir analogs as potent antiviral inhibitors

(2016) Zhao-Liang Yang et al.   TETRAHEDRON LETTERS

The formation of carbon–carbon and carbon–heteroatom bonds using silver tetrafluoroborate as a promoter

(2016) Matthew Chilaka Achilonu et al.   Arabian Journal of Chemistry

Investigating the Influence of (Deoxy)fluorination on the Lipophilicity of Non-UV-Active Fluorinated Alkanols and Carbohydrates by a New log P Determination Method

(2015) Bruno Linclau et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Catalytic Mechanism of Human Parainfluenza Virus Type 3 Haemagglutinin-Neuraminidase Revealed

(2015) Larissa Dirr et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Inhibitory efficiencies for mechanism-based inactivators of sialidases

(2015) Kobra Khazaei et al.   CANADIAN JOURNAL OF CHEMISTRY

Understanding viral neuraminidase inhibition by substituted difluorosialic acids

(2015) S. Weck et al.   CHEMICAL COMMUNICATIONS

Recent advances in the development of synthetic chemical probes for glycosidase enzymes

(2015) Helen M. Burke et al.   CHEMICAL COMMUNICATIONS

Monofluorination of Organic Compounds: 10 Years of Innovation

(2015) Pier Alexandre Champagne et al.   CHEMICAL REVIEWS

Recent Developments in Synthetic Carbohydrate-Based Diagnostics, Vaccines, and Therapeutics

(2015) Alberto Fernández-Tejada et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organofluorine chemistry: applications, sources and sustainability

(2015) Antal Harsanyi et al.   GREEN CHEMISTRY

Synthesis and antiviral evaluation of 2′,3′-dideoxy-2′,3′-difluoro-D-arabinofuranosyl 2,6-disubstituted purine nucleosides

(2015) Raymond F. Schinazi et al.   HETEROCYCLIC COMMUNICATIONS

The synthesis of tetrafluorinated aminosugars

(2015) Clément Q. Fontenelle et al.   JOURNAL OF FLUORINE CHEMISTRY

The synthesis of mono- and difluorinated 2,3-dideoxy-d-glucopyranoses

(2015) Lewis Mtashobya et al.   JOURNAL OF FLUORINE CHEMISTRY

Investigation and Conformational Analysis of Fluorinated Nucleoside Antibiotics Targeting Siderophore Biosynthesis

(2015) Surendra Dawadi et al.   JOURNAL OF ORGANIC CHEMISTRY

Toward a Molecular Lego Approach for the Diversity-Oriented Synthesis of Cyclodextrin Analogues Designed as Scaffolds for Multivalent Systems

(2015) Mathieu L. Lepage et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 2-deoxy-2,2-difluoro-α-maltosyl fluoride and its X-ray structure in complex with Streptomyces coelicolor GlgEI-V279S

(2015) Sandeep Thanna et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of Fluorosugar Reagents for the Construction of Well-Defined Fluoroglycoproteins

(2015) Míriam Salvadó et al.   ORGANIC LETTERS

Rules and Stereoelectronic Guidelines for the Anionic Nucleophilic Displacement of Furanoside and Furanose O-Sulfonates

(2015) Karl J. Hale et al.   ORGANIC LETTERS

Coordination diversity in hydrogen-bonded homoleptic fluoride–alcohol complexes modulates reactivity

(2015) Keary M. Engle et al.   Chemical Science

Glycan based Detection and Drug Susceptibility of Influenza Virus

(2014) Hieu Dinh et al.   ANALYTICAL CHEMISTRY

Tuning Mechanism-Based Inactivators of Neuraminidases: Mechanistic and Structural Insights

(2014) Sabrina Buchini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Structural Insight into How Streptomyces coelicolor Maltosyl Transferase GlgE Binds α-Maltose 1-Phosphate and Forms a Maltosyl-enzyme Intermediate

(2014) Karl Syson et al.   BIOCHEMISTRY

Glycomimetics versus Multivalent Glycoconjugates for the Design of High Affinity Lectin Ligands

(2014) Samy Cecioni et al.   CHEMICAL REVIEWS

Fluorinated Mechanism-Based Inhibitors: Common Themes and Recent Developments

(2014) Christina Tysoe et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Synthesis of Pyranonucleoside-6′-triphosphates through thecycloSal-Method

(2014) Johanna Huchting et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Exploring Human Parainfluenza Virus Type-1 Hemagglutinin–Neuraminidase as a Target for Inhibitor Discovery

(2014) Ibrahim M. El-Deeb et al.   JOURNAL OF MEDICINAL CHEMISTRY

Effects of Sugar Functional Groups, Hydrophobicity, and Fluorination on Carbohydrate–DNA Stacking Interactions in Water

(2014) Ricardo Lucas et al.   JOURNAL OF ORGANIC CHEMISTRY

Stereoselectivity of the Honda–Reformatsky Reaction in Reactions with Ethyl Bromodifluoroacetate with α-Oxygenated Sulfinylimines

(2014) Clément Q. Fontenelle et al.   JOURNAL OF ORGANIC CHEMISTRY

Rigid 2′,4′-Difluororibonucleosides: Synthesis, Conformational Analysis, and Incorporation into Nascent RNA by HCV Polymerase

(2014) Saúl Martínez-Montero et al.   JOURNAL OF ORGANIC CHEMISTRY

Phosphodiesters serve as potentially tunable aglycones for fluoro sugar inactivators of retaining β-glycosidases

(2014) B. P. Rempel et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

An Update of the Rules for Pyranoside Sulfonate Displacement

(2014) Karl J. Hale et al.   ORGANIC LETTERS

Structure-guided discovery of potent and dual-acting human parainfluenza virus haemagglutinin–neuraminidase inhibitors

(2014) Patrice Guillon et al.   Nature Communications

Investigating virus–glycan interactions using glycan microarrays

(2014) David F Smith et al.   Current Opinion in Virology

Intramolecular OH⋅⋅⋅FC Hydrogen Bonding in Fluorinated Carbohydrates: CHF is a Better Hydrogen Bond Acceptor than CF2

(2013) Guy T. Giuffredi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Introduction of Fluorine and Fluorine-Containing Functional Groups

(2013) Theresa Liang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

RCAI-61 and related 6′-modified analogs of KRN7000: Their synthesis and bioactivity for mouse lymphocytes to produce interferon-γ in vivo

(2013) Takuya Tashiro et al.   BIOORGANIC & MEDICINAL CHEMISTRY

The synthesis of a series of deoxygenated 2,3-difluoro-N-acteylneuraminic acid derivatives as potential sialidase inhibitors

(2013) Stefan Hader et al.   CARBOHYDRATE RESEARCH

Tetrafluorination of Sugars as Strategy for Enhancing Protein-Carbohydrate Affinity: Application to UDP-GalpMutase Inhibition

(2013) Inès N'Go et al.   CHEMISTRY-A EUROPEAN JOURNAL

Fluorinated Carbohydrates as Lectin Ligands: Dissecting Glycan-Cyanovirin Interactions by Using19F NMR Spectroscopy

(2013) Elena Matei et al.   CHEMISTRY-A EUROPEAN JOURNAL

Carbohydrate-Based Molecules for Molecular Imaging in Nuclear Medicine

(2013) Goreti Ribeiro Morais et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Short synthetic preparation of enantiomerically pure tetrafluoroethylenated sugar derivatives

(2013) Tsutomu Konno et al.   JOURNAL OF FLUORINE CHEMISTRY

Fluorosugars: An improved synthesis of the 2,3,4-trideoxy-2,3,4-trifluoro hexose analogue of d-glucose

(2013) Michael J. Corr et al.   JOURNAL OF FLUORINE CHEMISTRY

Cell-permeable probe for identification and imaging of sialidases

(2013) C.-S. Tsai et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Mechanism-Based Covalent Neuraminidase Inhibitors with Broad-Spectrum Influenza Antiviral Activity

(2013) J.-H. Kim et al.   SCIENCE

Structure and stereochemistry of an anti-inflammatory anhydrosugar from the Australian marine sponge Plakinastrella clathrata and the synthesis of two analogues

(2013) Peter L. Katavic et al.   TETRAHEDRON

Torsional control of stereoselectivities in electrophilic additions and cycloadditions to alkenes

(2013) Hao Wang et al.   Chemical Science

Multivalency as a Chemical Organization and Action Principle

(2012) Carlo Fasting et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of a fluorescently tagged sialic acid analogue useful for live-cell imaging

(2012) Katsuhiko Suzuki et al.   CHEMICAL COMMUNICATIONS

Conformational Analysis of Furanoside-Containing Mono- and Oligosaccharides

(2012) Hashem A. Taha et al.   CHEMICAL REVIEWS

Multivalent glycoconjugates as anti-pathogenic agents

(2012) Anna Bernardi et al.   CHEMICAL SOCIETY REVIEWS

Fluorine-Directed β-Galactosylation: Chemical Glycosylation Development by Molecular Editing

(2012) Estelle Durantie et al.   CHEMISTRY-A EUROPEAN JOURNAL

Fluorinated Carbohydrates as Lectin Ligands: Biorelevant Sensors with Capacity to Monitor Anomer Affinity in 19F-NMR-Based Inhibitor Screening

(2012) Sabine André et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Suite of Activity-Based Probes for Cellulose-Degrading Enzymes

(2012) Lacie M. Chauvigné-Hines et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The conformation of tetrafluorinated methyl galactoside anomers: crystallographic and NMR studies

(2011) Bruno Linclau et al.   CARBOHYDRATE RESEARCH

Facile synthesis of acacetin-7-O-β-d-galactopyranoside

(2011) James T. Zacharia et al.   CARBOHYDRATE RESEARCH

Activity-Based Profiling of Retaining β-Glucosidases: A Comparative Study

(2011) Martin D. Witte et al.   CHEMBIOCHEM

Synthesis of a MUC1-glycopeptide–BSA conjugate vaccine bearing the 3′-deoxy-3′-fluoro-Thomsen–Friedenreich antigen

(2011) Anja Hoffmann-Röder et al.   CHEMICAL COMMUNICATIONS

Antibody recognition of fluorinated MUC1 glycopeptide antigens

(2011) Thomas Oberbillig et al.   CHEMICAL COMMUNICATIONS

De Novo Synthesis of Racemic 4-Deoxy-4,4-difluoro- and 2,4-Dideoxy-2,4,4-trifluorohexosides

(2011) Guy T. Giuffredi et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Fluorinated Ketoheptoses as Specific Diagnostic Agents

(2011) Daniel Waschke et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Facile synthesis of 4-deoxy-4-fluoro-α-d-talopyranoside, 4-deoxy-4-fluoro-α-d-idopyranoside and 2,4-dideoxy-2,4-difluoro-α-d-talopyranoside

(2011) Guy T. Giuffredi et al.   JOURNAL OF FLUORINE CHEMISTRY

Stereoselective Synthesis of PSI-352938: A β-d-2′-Deoxy-2′-α-fluoro-2′-β-C-methyl-3′,5′-cyclic Phosphate Nucleotide Prodrug for the Treatment of HCV

(2011) P. Ganapati Reddy et al.   JOURNAL OF ORGANIC CHEMISTRY

Structural, Mechanistic, and Computational Analysis of the Effects of Anomeric Fluorines on Anomeric Fluoride Departure in 5-Fluoroxylosyl Fluorides

(2011) Seung Seo Lee et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Skeletal rearrangements resulting from reactions of 1,6:2,3- and 1,6:3,4-dianhydro-β-d-hexopyranoses with diethylaminosulphur trifluoride

(2011) Jindřich Karban et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

d-Gluco-hept-2-ulose and Novel Deoxyfluoro Derivatives as Seven-Carbon Analogues of F-Deoxy-d-glucose (FDG)

(2011) Joachim Thiem et al.   SYNTHESIS-STUTTGART

Two procedures for the syntheses of labeled sialic acids and their 1,7-lactones

(2011) Pietro Allevi et al.   TETRAHEDRON-ASYMMETRY

Synthetic Antitumor Vaccines from Tetanus Toxoid Conjugates of MUC1 Glycopeptides with the Thomsen-Friedenreich Antigen and a Fluorine-Substituted Analogue

(2010) Anja Hoffmann-Röder et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Fluorine-Directed Glycosylation

(2010) Christoph Bucher et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and in vitro antiviral activities of 3′-fluoro (or chloro) and 2′,3′-difluoro 2′,3′-dideoxynucleoside analogs against hepatitis B and C viruses

(2010) Naveen C. Srivastav et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Fluorosugars: synthesis of the 2,3,4-trideoxy-2,3,4-trifluoro hexose analogues of d-glucose and d-altrose and assessment of their erythrocyte transmembrane transport

(2010) Stefano Bresciani et al.   CHEMICAL COMMUNICATIONS

Fluorinated Glycosyl Amino Acids for Mucin-Like Glycopeptide Antigen Analogues

(2010) Sarah Wagner et al.   CHEMISTRY-A EUROPEAN JOURNAL

Recent Progress in Synthesis and Applications of Fluorinated Carbohydrates

(2010) Yuan Cheng et al.   CURRENT ORGANIC CHEMISTRY

Synthesis and Structure Elucidation of Benzoylated Deoxyfluoropyranosides

(2010) Aslan M. Esmurziev et al.   JOURNAL OF CARBOHYDRATE CHEMISTRY

Antiviral Activity of Various 1-(2′-Deoxy-β-d-lyxofuranosyl), 1-(2′-Fluoro-β-d-xylofuranosyl), 1-(3′-Fluoro-β-d-arabinofuranosyl), and 2′-Fluoro-2′,3′-didehydro-2′,3′-dideoxyribose Pyrimidine Nucleoside Analogues against Duck Hepatitis B Virus (DHBV) and Human Hepatitis B Virus (HBV) Replication

(2010) Naveen C. Srivastav et al.   JOURNAL OF MEDICINAL CHEMISTRY

Aminodifluorosulfinium Salts: Selective Fluorination Reagents with Enhanced Thermal Stability and Ease of Handling†,‡

(2010) Alexandre L’Heureux et al.   JOURNAL OF ORGANIC CHEMISTRY

Formation of Homooligosaccharides Using Base-Promoted Glycosylation of Unprotected Glycosyl Fluorides

(2010) Andreas Steinmann et al.   MACROMOLECULES

Synthesis and O-phosphorylation of 3,3,4,4-tetrafluoroaryl-C-nucleoside analogues

(2010) Laurent Bonnac et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of sulfonamide-based kinase inhibitors from sulfonates by exploiting the abrogated SN2 reactivity of 2,2,2-trifluoroethoxysulfonates

(2010) Christopher Wong et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Process Development of Selectively Benzoylated and Fluorinated Glycosyl Donors

(2010) Franz J. Weiberth et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Novel Introduction of a Tetrafluoroethylene (-CF2CF2-) Unit into Organic Molecules

(2010) Tsutomu Konno et al.   SYNTHESIS-STUTTGART

Metabolic Labeling of Sialic Acids in Living Animals with Alkynyl Sugars

(2009) Pamela V. Chang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Non-Stick Sugars: Synthesis of Difluorosugar Fluorides as Potential Glycosidase Inactivators

(2009) Brian P. Rempel et al.   AUSTRALIAN JOURNAL OF CHEMISTRY

d-Glucose- and d-mannose-based antimetabolites. Part 2. Facile synthesis of 2-deoxy-2-halo-d-glucoses and -d-mannoses

(2009) Izabela Fokt et al.   CARBOHYDRATE RESEARCH

Bacterial Adhesins in Host-Microbe Interactions

(2009) Kimberly A. Kline et al.   Cell Host & Microbe

Fluorinated Carbohydrates as Lectin Ligands: Versatile Sensors in19F-Detected Saturation Transfer Difference NMR Spectroscopy

(2009) Tammo Diercks et al.   CHEMISTRY-A EUROPEAN JOURNAL

Sweets for Catalysis - Facile Optimisation of Carbohydrate-Based Bis(oxazoline) Ligands

(2009) Tobias Minuth et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A regio- and stereoisomeric study of allylic alcohol fluorination with a range of reagents

(2009) Stefano Bresciani et al.   JOURNAL OF FLUORINE CHEMISTRY

An Efficient and Diastereoselective Synthesis of PSI-6130: A Clinically Efficacious Inhibitor of HCV NS5B Polymerase

(2009) Peiyuan Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

DAST-Mediated Regioselective Anomeric Group Migration in Saccharides

(2009) Po-Chiao Lin et al.   JOURNAL OF ORGANIC CHEMISTRY

From carbohydrate leads to glycomimetic drugs

(2009) Beat Ernst et al.   NATURE REVIEWS DRUG DISCOVERY

Synthesis and Antiviral Activity of Purine 2′,3′-Dideoxy-2′,3′-Difluoro-D-Arabinofuranosyl Nucleosides

(2009) Grigorii G. Sivets et al.   NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS

Enantioselective synthesis of tetrafluorinated ribose and fructose

(2009) Bruno Linclau et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Aminodifluorosulfinium Tetrafluoroborate Salts as Stable and Crystalline Deoxofluorinating Reagents

(2009) Francis Beaulieu et al.   ORGANIC LETTERS

A Highly Efficient Conversion of Primary or Secondary Alcohols into Fluorides with n-Perfluorobutanesulfonyl Fluoride-Tetrabutylammonium Triphenyldifluorosilicate

(2009) Xueqing Zhao et al.   SYNLETT

Direct synthesis of 1,6-anhydro sugars from unprotected glycopyranoses by using 2-chloro-1,3-dimethylimidazolinium chloride

(2009) Tomonari Tanaka et al.   TETRAHEDRON LETTERS

Tetrabutylammonium Tetra(tert-Butyl Alcohol)-Coordinated Fluoride as a Facile Fluoride Source

(2008) Dong Wook Kim et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A New Generation of SpecificTrypanosoma cruzi trans-Sialidase Inhibitors

(2008) Sabrina Buchini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Pasteurella multocida sialic acid aldolase: a promising biocatalyst

(2008) Yanhong Li et al.   APPLIED MICROBIOLOGY AND BIOTECHNOLOGY

Recent knowledge and innovations related to hexofuranosides: structure, synthesis and applications

(2008) Pauline Peltier et al.   CARBOHYDRATE RESEARCH

Stereospecific synthesis of sugar-1-phosphates and their conversion to sugar nucleotides

(2008) Shannon C. Timmons et al.   CARBOHYDRATE RESEARCH

Fragmentation of Carbohydrate Anomeric Alkoxyl Radicals: New Synthesis of Chiral 1-Fluoro-1-halo-1-iodoalditols

(2008) Cosme G. Francisco et al.   CHEMISTRY-A EUROPEAN JOURNAL

Covalent inhibitors of glycosidases and their applications in biochemistry and biology

(2008) B. P Rempel et al.   GLYCOBIOLOGY

Fluorinated nucleosides: Synthesis and biological implication

(2008) Peng Liu et al.   JOURNAL OF FLUORINE CHEMISTRY

Synthesis and Testing of 2-Deoxy-2,2-Dihaloglycosides as Mechanism-Based Inhibitors of α-Glycosidases

(2008) Ran Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Facile Nucleophilic Fluorination Reactions Usingtert-Alcohols as a Reaction Medium:  Significantly Enhanced Reactivity of Alkali Metal Fluorides and Improved Selectivity

(2008) Dong Wook Kim et al.   JOURNAL OF ORGANIC CHEMISTRY

Protein-glycan interactions in the control of innate and adaptive immune responses

(2008) Yvette van Kooyk et al.   NATURE IMMUNOLOGY

Enantioselective Synthesis of Tetrafluorinated Glucose and Galactose

(2008) Roxana S. Timofte et al.   ORGANIC LETTERS

A short synthesis of 4-deoxy-4-fluoroglucosaminides: Methylumbelliferyl N-acetyl-4-deoxy-4-fluoro-β-D-glucosaminide

(2008) N. A. Markina et al.   RUSSIAN JOURNAL OF BIOORGANIC CHEMISTRY

Synthesis and Use of Mechanism-Based Protein-Profiling Probes for Retaining β-d-Glucosaminidases Facilitate Identification ofPseudomonas aeruginosaNagZ

(2007) Keith A. Stubbs et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY